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Search Results for " glucocorticoid receptor agonist "

20

Compounds

Cat No. Product Name Synonyms Targets
T11417 Glucocorticoid receptor agonist Others
Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.
T37908 Glucocorticoid receptor agonist-1 Glucocorticoid Receptor
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1].
T74697 Glucocorticoid receptor agonist-2
Glucocorticoid receptor agonist-2 (compound 21), a glucocorticoid receptor agonist exhibiting an IC50 value of 6.6 nM, serves as an active reference for ABBV-3373 [1]. This compound is instrumental in the synthesis of an...
T74116 Glucocorticoid receptor agonist-1 Ala-Ala-Mal
Glucocorticoid receptor agonist-1 Ala-Ala-Mal (compound 88), a glucocorticosteroid and glucocorticoid receptor agonist, can be conjugated with Adalimumab to formulate an ADC [1].
T77869 Glucocorticoid receptor agonist-2 Ala-Ala-Mal
Glucocorticoid receptor agonist-2 Ala-Ala-Mal (compound 79) serves as a precursor for synthesizing anti-inflammatory antibody-drug conjugate (ADC) molecules and acts as an active reference for ABBV-3373 [1].
T75016 Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal
Glucocorticoid Receptor Agonist-1 Phosphate Ala-Ala-Mal functions as a glucocorticoid receptor agonist, utilized in the formulation of anti-CD40 antibody agent conjugates (ADC). It serves as a research tool for exploring...
T77835 Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Br
Glucocorticoid Receptor Agonist-1 Phosphate (Gly-Glu-Br) is an antibody-drug conjugate (ADC) linker utilized in the synthesis of ABBV-154, ABBV-927, ABBV-368, and related analogs [1].
T82303 Glucocorticoid receptor agonist-1 phosphate Gly-Glu TFA
Glucocorticoid Receptor Agonist-1 Phosphate Gly-Glu (TFA) serves as a cleavable linker for the synthesis of Antibody-Drug Conjugates (ADCs).
T75130 Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br
Glucocorticoid Receptor Agonist-1 Phosphate Ala-Ala-Br is a drug-linker conjugate for antibody-drug conjugates (ADCs), serving as a reaction reagent in the creation of anti-CD40 antibody agent conjugates [1].
T15102 Dexamethasone palmitate DXP Glucocorticoid Receptor
Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone, shows a 47-fold lower affinity for the glucocorticoid receptor than Dexamethasone. Dexamethasone palmitate is a glucocorticoid receptor agonist and an...
T1683 Actriol Epiestriol Glucocorticoid Receptor
Actriol (Epiestriol) is always used as Glucocorticoid Receptor agonist.
T0270 Hydrocortisone 17-butyrate Cortisol 17-butyrate,Hydrocortisone butyrate Glucocorticoid Receptor , Annexin A , Adrenergic Receptor
Hydrocortisone 17-butyrate (Cortisol 17-butyrate) is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects.
T22818 GSK9027 GR agonist 23a,GSK 9027,GSK-9027 Glucocorticoid Receptor
GSK9027 (GR agonist 23a) is a nonsteroidal glucocorticoid receptor (GR) agonist.GSK9027 is a partial agonist on the 2×GRE reporter gene compared to dexamethasone and is less active than dexamethasone activity.
T8396 Prednisone acetate Prednisone 21-acetate Glucocorticoid Receptor
Prednisone acetate (Prednisone 21-acetate) is a glucocorticoid receptor agonist with immunomodulating properties and anti-inflammatory.
T8777 Beclometasone BecloMethasone Glucocorticoid Receptor
Beclometasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma.
T15451 GW-870086 Glucocorticoid Receptor
GW-870086 is an effective anti-inflammatory agent. GW-870086 also plays a role in a glucocorticoid receptor agonist (pIC50: 10.1 in A549 cells expressing NF-κB).
T0188 Fluticasone (propionate) CCI-187881,Fluticasone propionate Glucocorticoid Receptor , Virus Protease , Estrogen/progestogen Receptor , Phospholipase , Endogenous Metabolite
Fluticasone propionate (CCI-187881), derived from fluticasone used to remedy asthma and allergic rhinitis, is a high affinity, selective GR (glucocorticoid receptor) agonist.
T1124 Flumethasone Flumetasone,RS-2177,NSC-54702 Glucocorticoid Receptor
Flumethasone (RS-2177) is a glucocorticoid receptor agonist, with anti-inflammatory, antipruritic and vasoconstrictive properties.
T1666 Fludrocortisone acetate 9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,9α-fluorocortisol acetate Glucocorticoid Receptor , Autophagy
Fludrocortisone acetate (9α-Fludrocortisone acetate) , a glucocorticoid-receptor agonist, binds to cytoplasmic receptors, translocates to the nucleus, and subsequently initiates the transcription of glucocorticoid-respon...
T1076 Dexamethasone MK 125,Prednisolone F,NSC 34521,Hexadecadrol Glucocorticoid Receptor , Mitophagy , IL Receptor , SARS-CoV , Antibacterial , Antibiotic , Autophagy , Complement System
Dexamethasone (Hexadecadrol) is a glucocorticoid receptor agonist and an IL receptor modulator. Dexamethasone has anti-inflammatory and immunosuppressive activity and induces autophagy. Dexamethasone inhibits LPS-induced...

Compounds

Glucocorticoid receptor agonist
T11417
Synonym:
Target: Others
Glucocorticoid receptor agonist-1
T37908
Synonym:
Target: Glucocorticoid Receptor
Glucocorticoid receptor agonist-2
T74697
Synonym:
Target:
Glucocorticoid receptor agonist-1 Ala-Ala-Mal
T74116
Synonym:
Target:
Glucocorticoid receptor agonist-2 Ala-Ala-Mal
T77869
Synonym:
Target:
Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal
T75016
Synonym:
Target:
Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Br
T77835
Synonym:
Target:
Glucocorticoid receptor agonist-1 phosphate Gly-Glu TFA
T82303
Synonym:
Target:
Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br
T75130
Synonym:
Target:
Dexamethasone palmitate
T15102
Synonym: DXP
Target: Glucocorticoid Receptor
Actriol
T1683
Synonym: Epiestriol
Target: Glucocorticoid Receptor
Hydrocortisone 17-butyrate
T0270
Synonym: Cortisol 17-butyrate,Hydrocortisone butyrate
Target: Glucocorticoid Receptor, Annexin A, Adrenergic Receptor
GSK9027
T22818
Synonym: GR agonist 23a,GSK 9027,GSK-9027
Target: Glucocorticoid Receptor
Prednisone acetate
T8396
Synonym: Prednisone 21-acetate
Target: Glucocorticoid Receptor
Beclometasone
T8777
Synonym: BecloMethasone
Target: Glucocorticoid Receptor
GW-870086
T15451
Synonym:
Target: Glucocorticoid Receptor
Fluticasone (propionate)
T0188
Synonym: CCI-187881,Fluticasone propionate
Target: Glucocorticoid Receptor, Virus Protease, Estrogen/progestogen Receptor, Phospholipase, Endogenous Metabolite
Flumethasone
T1124
Synonym: Flumetasone,RS-2177,NSC-54702
Target: Glucocorticoid Receptor
Fludrocortisone acetate
T1666
Synonym: 9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,9α-fluorocortisol acetate
Target: Glucocorticoid Receptor, Autophagy
Dexamethasone
T1076
Synonym: MK 125,Prednisolone F,NSC 34521,Hexadecadrol
Target: Glucocorticoid Receptor, Mitophagy, IL Receptor, SARS-CoV, Antibacterial, Antibiotic, Autophagy, Complement System
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TargetMol