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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T11417 | Glucocorticoid receptor agonist | Others | |
Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist. | |||
T37908 | Glucocorticoid receptor agonist-1 | Glucocorticoid Receptor | |
Glucocorticoid receptor agonist-1 is a potent glucocorticoid receptor agonist with an IC50 of 2.8 nM[1]. | |||
T74697 | Glucocorticoid receptor agonist-2 | ||
Glucocorticoid receptor agonist-2 (compound 21), a glucocorticoid receptor agonist exhibiting an IC50 value of 6.6 nM, serves as an active reference for ABBV-3373 [1]. This compound is instrumental in the synthesis of an... | |||
T74116 | Glucocorticoid receptor agonist-1 Ala-Ala-Mal | ||
Glucocorticoid receptor agonist-1 Ala-Ala-Mal (compound 88), a glucocorticosteroid and glucocorticoid receptor agonist, can be conjugated with Adalimumab to formulate an ADC [1]. | |||
T77869 | Glucocorticoid receptor agonist-2 Ala-Ala-Mal | ||
Glucocorticoid receptor agonist-2 Ala-Ala-Mal (compound 79) serves as a precursor for synthesizing anti-inflammatory antibody-drug conjugate (ADC) molecules and acts as an active reference for ABBV-3373 [1]. | |||
T75016 | Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal | ||
Glucocorticoid Receptor Agonist-1 Phosphate Ala-Ala-Mal functions as a glucocorticoid receptor agonist, utilized in the formulation of anti-CD40 antibody agent conjugates (ADC). It serves as a research tool for exploring... | |||
T77835 | Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Br | ||
Glucocorticoid Receptor Agonist-1 Phosphate (Gly-Glu-Br) is an antibody-drug conjugate (ADC) linker utilized in the synthesis of ABBV-154, ABBV-927, ABBV-368, and related analogs [1]. | |||
T82303 | Glucocorticoid receptor agonist-1 phosphate Gly-Glu TFA | ||
Glucocorticoid Receptor Agonist-1 Phosphate Gly-Glu (TFA) serves as a cleavable linker for the synthesis of Antibody-Drug Conjugates (ADCs). | |||
T75130 | Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Br | ||
Glucocorticoid Receptor Agonist-1 Phosphate Ala-Ala-Br is a drug-linker conjugate for antibody-drug conjugates (ADCs), serving as a reaction reagent in the creation of anti-CD40 antibody agent conjugates [1]. | |||
T15102 | Dexamethasone palmitate | DXP | Glucocorticoid Receptor |
Dexamethasone palmitate (DXP), a lipophilic prodrug of Dexamethasone, shows a 47-fold lower affinity for the glucocorticoid receptor than Dexamethasone. Dexamethasone palmitate is a glucocorticoid receptor agonist and an... | |||
T1683 | Actriol | Epiestriol | Glucocorticoid Receptor |
Actriol (Epiestriol) is always used as Glucocorticoid Receptor agonist. | |||
T0270 | Hydrocortisone 17-butyrate | Cortisol 17-butyrate,Hydrocortisone butyrate | Glucocorticoid Receptor , Annexin A , Adrenergic Receptor |
Hydrocortisone 17-butyrate (Cortisol 17-butyrate) is a synthetic glucocorticoid receptor agonist with antiinflammatory, antipruritic and vasoconstrictive effects. | |||
T22818 | GSK9027 | GR agonist 23a,GSK 9027,GSK-9027 | Glucocorticoid Receptor |
GSK9027 (GR agonist 23a) is a nonsteroidal glucocorticoid receptor (GR) agonist.GSK9027 is a partial agonist on the 2×GRE reporter gene compared to dexamethasone and is less active than dexamethasone activity. | |||
T8396 | Prednisone acetate | Prednisone 21-acetate | Glucocorticoid Receptor |
Prednisone acetate (Prednisone 21-acetate) is a glucocorticoid receptor agonist with immunomodulating properties and anti-inflammatory. | |||
T8777 | Beclometasone | BecloMethasone | Glucocorticoid Receptor |
Beclometasone is a prototype glucocorticoid receptor agonist. It is used topically as an anti-inflammatory agent and in aerosol form for the treatment of asthma. | |||
T15451 | GW-870086 | Glucocorticoid Receptor | |
GW-870086 is an effective anti-inflammatory agent. GW-870086 also plays a role in a glucocorticoid receptor agonist (pIC50: 10.1 in A549 cells expressing NF-κB). | |||
T0188 | Fluticasone (propionate) | CCI-187881,Fluticasone propionate | Glucocorticoid Receptor , Virus Protease , Estrogen/progestogen Receptor , Phospholipase , Endogenous Metabolite |
Fluticasone propionate (CCI-187881), derived from fluticasone used to remedy asthma and allergic rhinitis, is a high affinity, selective GR (glucocorticoid receptor) agonist. | |||
T1124 | Flumethasone | Flumetasone,RS-2177,NSC-54702 | Glucocorticoid Receptor |
Flumethasone (RS-2177) is a glucocorticoid receptor agonist, with anti-inflammatory, antipruritic and vasoconstrictive properties. | |||
T1666 | Fludrocortisone acetate | 9α-Fluorcortisol acetate,9α-Fludrocortisone acetate,9α-fluorocortisol acetate | Glucocorticoid Receptor , Autophagy |
Fludrocortisone acetate (9α-Fludrocortisone acetate) , a glucocorticoid-receptor agonist, binds to cytoplasmic receptors, translocates to the nucleus, and subsequently initiates the transcription of glucocorticoid-respon... | |||
T1076 | Dexamethasone | MK 125,Prednisolone F,NSC 34521,Hexadecadrol | Glucocorticoid Receptor , Mitophagy , IL Receptor , SARS-CoV , Antibacterial , Antibiotic , Autophagy , Complement System |
Dexamethasone (Hexadecadrol) is a glucocorticoid receptor agonist and an IL receptor modulator. Dexamethasone has anti-inflammatory and immunosuppressive activity and induces autophagy. Dexamethasone inhibits LPS-induced... |